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Bremelanotide acetate

CAS No. 1607799-13-2

Bremelanotide acetate( PT-141 acetate )

Catalog No. M12310 CAS No. 1607799-13-2

Bremelanotide acetate is an analogue of the naturally occurring peptide alpha-MSH; melanocortin receptor agonist.

Purity : >98% (HPLC)

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Biological Information

  • Product Name
    Bremelanotide acetate
  • Note
    Research use only, not for human use.
  • Brief Description
    Bremelanotide acetate is an analogue of the naturally occurring peptide alpha-MSH; melanocortin receptor agonist.
  • Description
    Bremelanotide acetate is an analogue of the naturally occurring peptide alpha-MSH; melanocortin receptor agonist.Sexual Dysfunction Phase 3 Clinical(In Vivo):Bremelanotide Acetate (50-200 μg/kg; s.c.; once) significantly increases proceptive solicitations in females primed with Estradiol benzoate+Progesterone or Estradiol benzoate alone in bilevel chambers.
  • In Vitro
    ——
  • In Vivo
    Bremelanotide Acetate (50-200 μg/kg; s.c.; once) significantly increases proceptive solicitations in females primed with Estradiol benzoate+Progesterone or Estradiol benzoate alone in bilevel chambers. Animal Model:Ovariectomized Long–Evans rats Dosage:50, 100, 200 μg/kg Administration:s.c.; once Result:Significantly increased proceptive solicitations in females primed with Estradiol benzoate+Progesterone or Estradiol benzoate alone in bilevel chambers.
  • Synonyms
    PT-141 acetate
  • Pathway
    GPCR/G Protein
  • Target
    Melanocortin Receptor
  • Recptor
    Melanocortin Receptor
  • Research Area
    Endocrinology
  • Indication
    Sexual Dysfunction

Chemical Information

  • CAS Number
    1607799-13-2
  • Formula Weight
    1085.215
  • Molecular Formula
    C52H72N14O12
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: ≥ 36 mg/mL
  • SMILES
    CCCCC(C(=O)NC1CC(=O)NCCCCC(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC1=O)CC2=CN=CN2)CC3=CC=CC=C3)CCCN=C(N)N)CC4=CNC5=CC=CC=C54)C(=O)O)NC(=O)C.CC(=O)O
  • Chemical Name
    (3S,6S,9R,12S,15S,23S)-12-((1H-imidazol-5-yl)methyl)-3-((1H-indol-3-yl)methyl)-15-((S)-2-acetamidohexanamido)-9-benzyl-6-(3-guanidinopropyl)-2,5,8,11,14,17-hexaoxo-1,4,7,10,13,18-hexaazacyclotricosane-23-carboxylic acid with acetic acid (1:1)

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Pfaus J, et al. J Sex Med. 2007 Nov;4 Suppl 4:269-79. 2. White WB, et al. J Hypertens. 2017 Apr;35(4):761-768.
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